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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T36057 Diallyl Tetrasulfide

ICD-1585

Diallyl tetrasulfide is an organosulfur compound that has been found in A. sativum and has diverse biological activities, including antimicrobial, antioxidant, and anticancer properties.[1],[2],[3],[4] It is active against the bacteria S. aureus and methicillin-resistant S. aureus (MRSA; MICs = 0.5 and 2 mg/L, respectively), as well as the fungi C. albicans, C. krusei, C. glabrata, A. niger, A. flavus, and A. fumigatus (MICs = 0.5, 4, 2, 1, 2, and 4 mg/L, respectively).[1] It reduces cadmium-ind...
T8238 Fosamprenavir Calcium Salt

福沙那伟钙,Diallyl Trisulfide,GW433908G

HIV Protease Microbiology/Virology; Proteases/Proteasome
Fosamprenavir Calcium Salt (GW433908G) 是抗逆转录病毒蛋白酶抑制剂 Amprenavir 的磷酸酯前药,具有改善的溶解性和抗HIV 感染作用。

化合物

Diallyl Tetrasulfide
Cat.No: T36057
Synonym: ICD-1585
Target:
Fosamprenavir Calcium Salt
Cat.No: T8238
Synonym: 福沙那伟钙,Diallyl Trisulfide,GW433908G
Target: HIV Protease
Cat. No. Product Name Target Signaling Pathways
TN1576 Diallyl disulfide

IL Receptor; NOS; NF-κB Immunology/Inflammation; NF-κB
Diallyl disulfide 能够抑制人角鲨烯单加氧酶,抑制角鲨烯环氧化的 IC50为 400 μM。它也具有抗肿瘤作用,同miR-200b 和miR-22联合使用可增强该作用。
T8693 Diallyl Trisulfide

二烯丙基三硫化物,二烯丙基三硫醚

Apoptosis; Reactive Oxygen Species; Antifungal Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Diallyl Trisulfide 是一种在大蒜中发现的有机多硫化物,可作为 H2S 供体。它抑制扩张性青霉的生长,有抗癌能力。

天然产物

Diallyl disulfide
Cat.No: TN1576
Synonym:
Target: IL Receptor, NOS, NF-κB
Diallyl Trisulfide
Cat.No: T8693
Synonym: 二烯丙基三硫化物,二烯丙基三硫醚
Target: Apoptosis, Reactive Oxygen Species, Antifungal
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